Chandana, P.; Nayyar, A. R.; Jain, R. Trityl-directed regiospecific synthesis of 2,3-disubstituted bioimidazoles. Syn. Comm. 2003 (in press).

Jain, R. Recent advancements in antimalarial drug development. Curr. Res. Inform. Pharm. Sci. 2002, 3, 2-8.

Jain, R.; Suryanarayana V.; Jain, M.; Kaur, N.; Singh, S.; Singh, P. P. Antimalarial activities of ring-substituted bioimidazoles. Bioorg. Med. Chem. Lett. 2002, 12, 1701-1704.

Jain, R.; Singh, J.; Perlman, J. H.; Gershengorn, M. C. Synthesis and biology of new thyrotropin-releasing hormone (TRH) analogues. Bioorg. Med. Chem. 2002, 10, 189-194.

Naraynan, S.; Suryanarayana V.; Jain, R. Regiospecific synthesis of 2,3-disubstituted-L-histidines and histamines. Bioorg. Med. Chem. Lett. 2001, 11, 1133-1136.

Jain, R. Convenient N-protection of L-pyroglutamic acid esters. Org. Prep. Proc. Intl. 2001, 33, 406-409.

Jain, R.; Balasubramanian V.; Nayyar, A. R.; Palde, P. B.; Jain, M.; Sachdeva, S.; Kaur, S.; Misra, V.; Singh, P. P.; Kaul, C. L. Ring-substituted quinolines as anti-tuberculosis agents. 2002, WTO Indian patent application no. 628/DEL/2002.

Jain, R.; Suryanarayana V.; Singh, P. P.; Kinhikar, A. G.; Singh, S.; Jain, M.; Sachdeva, S.; Misra, V.; Ramarao, P.; Kaul, C. L. Quinoline analogues with broad-spectrum of antimalarial activities. 2002, WTO Indian patent application no. 1112/DEL/2002.

Jain, R.; Hocart, S. J.; Murphy, W. A.; Taylor, J. E.; Coy, D. H. Highly potent cyclic disulfide antagonists of samatostatin. J. Med. Chem., 1999, 42, 1863-1871.

Jain, R.; Coy, D. H.; Murphy, W. A.; Rossowski, W. J.; Hocart. S. J.; Fuselier, J.; Taylor, J. E. Samatostatin receptor antagonist based on a mixed neuromedin B antagonist/samatostatin agonist. In Peptides: Frontiers of Peptide Science, Proceedings of the 15th American Peptide Symposium; Tam, J.P.; Kaumaya, P.T.P., Eds.; Kluwer: Dordrecht, The Netherlands, 1999; pp 526-529.

Jain, R.; Hocart, S. J.; Murphy, W. A.; Taylor, J. E.; Morgan, B.; Coy, D. H. Potent antagonists of samatostatin: Synthesis and biology. J. Med. Chem., 1998, 41, 1146-1154.

Jain, R., Avramovitch, B.; Cohen, L. A. Synthesis of ring-halogenated histidines and histamines. Tetrahedron, 1998, 54, 3235-3242.

Perlman, J. H.; Colson, A. O.; Jain, R.; Czyzewski, B.; Cohen, L. A.; Osman, R.; Gershengorn, M. C. Role of the extracellular loops of the thyrotropin-releasing hormone receptor: Evidence for an initial interaction with thyrotropin-releasing hormone. Biochemistry, 1997, 36, 15670-15676.

Jain, R.; Cohen, L. A.; King, M. M. Synthesis of novel ring-substituted histidines and histamines. Tetrahedron, 1997, 53, 4539-4548. 15) Jain, R.; El-Kadi, N.; King, M. M.; Cohen, L. A. Regiospecific alkylation of histidines and histamines at C-2. Tetrahedron, 1997, 53, 2365-2370.

Jain, R.; Cohen, L. A. Regiospecific alkylation of histidines and histamines at N-1(t). Tetrahedron, 1996, 52, 5363-5370.

Jain, R.; Siddiqi, S. M.; Ji, Xiao-duo; Melman, N.; Olah, M. E.; Evans, P.; Glashofer, M.; Padgett, W.; Cohen, L. A.; Daly, J. W.; Stiles, G.; Jacobson, K. A. A survey of non-xanthine derivatives as adenosine receptor ligands. Nucleosides Nucleotides, 1996, 15, 693-718.

Jain, R.; El-Kadi, N.; King, M. M.; Cohen, L. A. Synthesis of 2-substituted histidines and histamines. Peptides 1996, The Royal Society of Chemistry Perkin Division and The European Peptide Society, 24th Symposium of the European Peptide Society, Edinburgh, Scotland, 1996, Sept. 8-13 No. 96, page 309-310.